小針 良仁 Yoshihito Kohari

学位

学歴

職歴

担当授業科目（学部）

安全工学概論　地球環境, 安全工学概論　地域未来, 先端材料物質工学概論　地球環境（2020年度以前入学）, 先端材料物質総合工学I　先端材料, 先端材料物質総合工学II　先端材料, 科学技術英語　先端材料, 有機構造解析　先端材料, 先端材料物質工学演習　先端材料, 文献ゼミナール　先端材料, 工学基礎実験および演習 地球環境/短期履修, オホーツク地域と環境　地球環境, オホーツク地域と環境　地域未来

専門分野

有機合成化学, 不斉合成

研究テーマ

有機分子触媒を用いる不斉合成反応の開発

研究内容キーワード

有機分子触媒, 不斉合成, 生物活性化合物

所属学会

日本化学会, 有機合成化学協会

学術論文

論文名／掲載誌名等		掲載年月
A novel chiral oxazolidine organocatalyst for the synthesis of an oseltamivir intermadiate using a highly enantioselective Diels-Alder reaction of 1,2-dihydropyridine Chem. Commun., 46, 26, 4827-4829		2010-05
Efficient synthetic methodology of biflavones having a ring-a ring of two flavone units using Suzuki cross-coupling reactions Heterocycles, 81, 8, 1871-1879		2010-06
Efficient synthetic methodology of flav-3-enes using reductive elimination of flav-4-triflate Heterocycles, 82, 1, 843-850		2010-06
A highly enantioselective Diels Alder reaction of 1,2-dihydropyridine using a simple β-amino alcohol organocatalyst for a practical synthetic methodology of oseltamivir intermediate Tetrahedron Lett., 52, 37, 4745-4748		2011-09
Asymmetric synthesis of isoquinuclidines by Diels–Alder reaction of 1,2-dihydropyridine utilizing a chiral Lewis acid catalyst Tetrahedoron, 68, 6, 1774-1781		2012-02
キラルオキサゾリジン類を用いた触媒的不斉合成反応の開発 有機合成化学協会誌, 70, 2, 142-153		2012-02
One Step Synthesis of Optically Active Diazabicyclo[3.3.0]octanones or Diazabicyclo[4.3.0]nonanones by Asymmetric Conjugate Addition of Cyclic Hydrazine Heterocycles, 85, 5, 1045		2012-05
Highly Enantioselective Synthesis of Isoquinuclidine by Diels-Alder Reaction of 1,2-Dihydropyridine Utilizing Chiral Bisoxazoline-Cu(II) Complex Heterocycles, 86, 1, 203-217		2012-06
Asymmetric Synthesis of Isoquinuclidine by Diels-Alder Reaction of 1,2-Dihydropyridine and Chiral Dienophile Utilizing a Chiral Lewis Acid Heterocycles, 84, 1, 377-384		2012-06
CHIRAL PRIMARY AMINO SILYL ETHER ORGANOCATALYST FOR THE ENANTIOSELECTIVE DIELS-ALDER REACTION OF 1,2-DIHYDROPYRIDINES WITH AlDEHYDES Heterocycles, 86, 2		2012-08
Development of a Novel Method for Warfarin Synthesis via Lipase-Catalyzed Steroselective Michael Reaction Heterocycles, 87, 6, 1269-1278		2013-05
Enantioselective Diels–Alder Reaction of 1,2-Dihydropyridines with Aldehydes Using β-Amino Alcohol Organocatalyst J. Org. Chem., 79, 20, 9500-9511		2014-10
Chiral Primary Amino Amide Alcohol Organocatalyst for the Asymmetric Michael Addition of 4-Hydroxycoumarin with α,β-Unsaturated Ketones Heterocycles, 90, 2, 1124-1134		2015-07
Lipase-catalyzed domino Michael–aldol reaction of 2-methyl-1,3-cycloalkanedione and methyl vinyl ketone for the synthesis of bicyclic compounds Synth. commun., 46, 1, 46 - 54		2015-09
Silyloxy Amino Alcohol Organocatalyst for Enantioselective 1,3-Dipolar Cycloaddition of Nitrones to α,β-Unsaturated Aldehydes Eur. J. Org. Chem., 2015, 33, 7292-7300		2015-11
Chiral primary amino alcohol organobase catalysts for the asymmetric Diels–Alder reactions of anthrones with maleimides Tetrahedron: asymmetry, 26, 24, 1423-1429		2015-12
イミノ基により架橋した分解性ポリ(アルキルビニルエーテル)ゴムの合成 高分子論文集, 73, 73, 213-220		2016-03
Synthesis of Dibenzosiloles via Platinum-catalyzed Intramolecular Dehydrogenative Cyclization of 2-(Dialkylsilyl)biaryls Chemistry Letters, 45, 8, 857-859		2016-05
Simple Primary Amino Amide Organocatalyst for Enantioselective Aldol Reactions of Isatins with Ketones European Journal of Organic Chemistry, 2016, 22, 3748		2016-07
Site‐Selective Aliphatic C−H Silylation of 2‐Alkyloxazolines Catalyzed by Ruthenium Complexes CHEMCATCHEM, 8, 2202-2205		2016-07
Ruthenium-Catalysed Dehydrogenative C–H Borylation of Arenes with Pinacolborane Journal of Chemical Research, 40, 7, 393-396		2016-07
Rhodium(I)-Catalyzed Silylation of Aryl Iodides with Di(2-furyl)methylsilane Heterocycles, 95, 1, 152-157		2016-12
Simple primary β-amino alcohol catalyzed enantioselective Diels-Alder reaction of 3-hydroxy-2-pyridones Tetrahedron Letters, 57, 51, 5771		2016-12
Utilization of the Japanese peppermint herbal water byproduct of steam distillation as an antimicrobial agent Journal of Oleo Science, 67, 10, 1227-1233		2018-10
Unnatural tripeptide as highly enantioselective organocatalyst for asymmetric aldol reaction of isatins Tetrahedron Letters, 60, 5, 415-418		2018-12
Characteristics of Japanese Mint Extracts Obtained by Subcritical-water Treatment Food Science and Technology Research, 25, 5, 695-703		2019-01
Tripeptide-catalyzed Asymmetric Aldol Reaction of Trifluoromethylated Aromatic Ketones with Acetone Heterocycles, 99, 2, 841-847		2019-02
Preparation of monodisperse fully aromatic polyimide particles via the polycondensation of diethyl hexafluoroisopropylidenediphthalate with 4,4′-diaminodiphenylether in ethylene glycol Polymer Journal, 51, 405-412		2019-03
Tripeptide-Catalyzed Asymmetric Aldol Reaction Between α-ketoesters and Acetone Under Acidic Cocatalyst-Free Conditions Catalysts, 9, 6, 514		2019-06
Hydrodistillation by Solvent-Free Microwave Extraction of Fresh Japanese Peppermint (Mentha arvensis L.) Journal of Essential Oil Bearing Plants		2020-02
Conversion and Hydrothermal Decomposition of Major Components of Mint Essential Oil by Small-Scale Subcritical Water Treatment molecules, 25, 8, 1953		2020-04
トリペプチド触媒による活性化ケトン類の直接的不斉アルドール反応 有機合成化学協会誌, 78, 12, 1174-1183		2020-12
Organocatalyzed Asymmetric Aldol Reaction of α-Keto Amides with A Tripeptide Catalyst Synlett		2021-02

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