小針 良仁 Yoshihito Kohari

研究者情報
職名 助教
所属 地球環境工学科 - 先端材料物質工学コース
電話番号 0157-46-9440
メールアドレス kohari@mail.kitami-it.ac.jp
関連ウェブサイト http://www.mtrl.kitami-it.ac.jp/~murata/index.html
学位・学歴・職歴

学位

博士(工学) フラボノイド類の新規合成法の開発 2011

学歴

2003.3 室蘭工業大学工学部応用化学科卒業
2005.3 室蘭工業大学大学院工学研究科博士前期課程応用化学専攻修了
2011.3 室蘭工業大学大学院工学研究科博士後期課程物質工学専攻修了

職歴

2011.5-2015.3 室蘭工業大学大学院工学研究科博士研究員
2015.4-2016.3 北見工業大学マテリアル工学科特任助教
2016.4- 北見工業大学マテリアル工学科助教
担当科目・専門分野等
担当授業科目(学部)
文献ゼミナール マテ, 先端材料工学 マテ, 工学基礎実験および演習 地域未来/短期履修
専門分野
有機合成化学, 不斉合成
研究テーマ
有機分子触媒を用いる不斉合成反応の開発
研究内容キーワード
有機分子触媒, 不斉合成, 生物活性化合物
所属学会
日本化学会, 有機合成化学協会
学術論文等

学術論文

論文名/掲載誌名等   掲載年月
A novel chiral oxazolidine organocatalyst for the synthesis of an oseltamivir intermadiate using a highly enantioselective Diels-Alder reaction of 1,2-dihydropyridine
Chem. Commun., 46, 26, 4827-4829
2010-05
Efficient synthetic methodology of biflavones having a ring-a ring of two flavone units using Suzuki cross-coupling reactions
Heterocycles, 81, 8, 1871-1879
2010-06
Efficient synthetic methodology of flav-3-enes using reductive elimination of flav-4-triflate
Heterocycles, 82, 1, 843-850
2010-06
A highly enantioselective Diels Alder reaction of 1,2-dihydropyridine using a simple β-amino alcohol organocatalyst for a practical synthetic methodology of oseltamivir intermediate
Tetrahedron Lett., 52, 37, 4745-4748
2011-09
キラルオキサゾリジン類を用いた触媒的不斉合成反応の開発
有機合成化学協会誌, 70, 2, 142-153
2012-02
Asymmetric synthesis of isoquinuclidines by Diels–Alder reaction of 1,2-dihydropyridine utilizing a chiral Lewis acid catalyst
Tetrahedoron, 68, 6, 1774-1781
2012-02
One Step Synthesis of Optically Active Diazabicyclo[3.3.0]octanones or Diazabicyclo[4.3.0]nonanones by Asymmetric Conjugate Addition of Cyclic Hydrazine
Heterocycles, 85, 5, 1045
2012-05
Highly Enantioselective Synthesis of Isoquinuclidine by Diels-Alder Reaction of 1,2-Dihydropyridine Utilizing Chiral Bisoxazoline-Cu(II) Complex
Heterocycles, 86, 1, 203-217
2012-06
Asymmetric Synthesis of Isoquinuclidine by Diels-Alder Reaction of 1,2-Dihydropyridine and Chiral Dienophile Utilizing a Chiral Lewis Acid
Heterocycles, 84, 1, 377-384
2012-06
CHIRAL PRIMARY AMINO SILYL ETHER ORGANOCATALYST FOR THE ENANTIOSELECTIVE DIELS-ALDER REACTION OF 1,2-DIHYDROPYRIDINES WITH AlDEHYDES
Heterocycles, 86, 2
2012-08
Development of a Novel Method for Warfarin Synthesis via Lipase-Catalyzed Steroselective Michael Reaction
Heterocycles, 87, 6, 1269-1278
2013-05
Enantioselective Diels–Alder Reaction of 1,2-Dihydropyridines with Aldehydes Using β-Amino Alcohol Organocatalyst
J. Org. Chem., 79, 20, 9500-9511
2014-10
Chiral Primary Amino Amide Alcohol Organocatalyst for the Asymmetric Michael Addition of 4-Hydroxycoumarin with α,β-Unsaturated Ketones
Heterocycles, 90, 2, 1124-1134
2015-07
Lipase-catalyzed domino Michael–aldol reaction of 2-methyl-1,3-cycloalkanedione and methyl vinyl ketone for the synthesis of bicyclic compounds
Synth. commun., 46, 1, 46 - 54
2015-09
Silyloxy Amino Alcohol Organocatalyst for Enantioselective 1,3-Dipolar Cycloaddition of Nitrones to α,β-Unsaturated Aldehydes
Eur. J. Org. Chem., 2015, 33, 7292-7300
2015-11
Chiral primary amino alcohol organobase catalysts for the asymmetric Diels–Alder reactions of anthrones with maleimides
Tetrahedron: asymmetry, 26, 24, 1423-1429
2015-12
イミノ基により架橋した分解性ポリ(アルキルビニルエーテル)ゴムの合成
高分子論文集, 73, 73, 213-220
2016-03
Synthesis of Dibenzosiloles via Platinum-catalyzed Intramolecular Dehydrogenative Cyclization of 2-(Dialkylsilyl)biaryls
Chemistry Letters, 45, 8, 857-859
2016-05
Ruthenium-Catalysed Dehydrogenative C–H Borylation of Arenes with Pinacolborane
Journal of Chemical Research, 40, 7, 393-396
2016-07
Site‐Selective Aliphatic C−H Silylation of 2‐Alkyloxazolines Catalyzed by Ruthenium Complexes
CHEMCATCHEM, 8, 2202-2205
2016-07
Simple Primary Amino Amide Organocatalyst for Enantioselective Aldol Reactions of Isatins with Ketones
European Journal of Organic Chemistry, 2016, 22, 3748
2016-07
Rhodium(I)-Catalyzed Silylation of Aryl Iodides with Di(2-furyl)methylsilane
Heterocycles, 95, 1, 152-157
2016-12
Simple primary β-amino alcohol catalyzed enantioselective Diels-Alder reaction of 3-hydroxy-2-pyridones
Tetrahedron Letters, 57, 51, 5771
2016-12
Utilization of the Japanese peppermint herbal water byproduct of steam distillation as an antimicrobial agent
Journal of Oleo Science, 67, 10, 1227-1233
2018-10
Unnatural tripeptide as highly enantioselective organocatalyst for asymmetric aldol reaction of isatins
Tetrahedron Letters, 60, 5, 415-418
2018-12
Tripeptide-catalyzed Asymmetric Aldol Reaction of Trifluoromethylated Aromatic Ketones with Acetone
Heterocycles, 99, 2, 841-847
2019-02
Preparation of monodisperse fully aromatic polyimide particles via the polycondensation of diethyl hexafluoroisopropylidenediphthalate with 4,4′-diaminodiphenylether in ethylene glycol
Polymer Journal, 51, 405-412
2019-03