小針 良仁 Yoshihito Kohari

学位

学歴

職歴

担当授業科目（学部）

工学基礎実験および演習 地球環境/短期履修, 先端材料物質総合工学I　先端材料, 先端材料物質工学実験I　先端材料, 先端材料物質総合工学II　先端材料, 科学技術英語　先端材料, 有機構造解析　先端材料, 有機合成化学　先端材料, 文献ゼミナール　先端材料, オホーツク地域と環境　地球環境, オホーツク地域と環境　地域未来, 安全工学概論　地球環境, 安全工学概論　地域未来

専門分野

有機合成化学, 不斉合成

研究テーマ

有機分子触媒を用いる不斉合成反応の開発

研究内容キーワード

有機分子触媒, 不斉合成, 生物活性化合物

所属学会

日本化学会, 有機合成化学協会

学術論文

論文名／掲載誌名等		掲載年月
A novel chiral oxazolidine organocatalyst for the synthesis of an oseltamivir intermadiate using a highly enantioselective Diels-Alder reaction of 1,2-dihydropyridine Chem. Commun., 46, 26, 4827-4829		2010-05
Efficient synthetic methodology of biflavones having a ring-a ring of two flavone units using Suzuki cross-coupling reactions Heterocycles, 81, 8, 1871-1879		2010-06
Efficient synthetic methodology of flav-3-enes using reductive elimination of flav-4-triflate Heterocycles, 82, 1, 843-850		2010-06
A highly enantioselective Diels Alder reaction of 1,2-dihydropyridine using a simple β-amino alcohol organocatalyst for a practical synthetic methodology of oseltamivir intermediate Tetrahedron Lett., 52, 37, 4745-4748		2011-09
Asymmetric synthesis of isoquinuclidines by Diels–Alder reaction of 1,2-dihydropyridine utilizing a chiral Lewis acid catalyst Tetrahedoron, 68, 6, 1774-1781		2012-02
キラルオキサゾリジン類を用いた触媒的不斉合成反応の開発 有機合成化学協会誌, 70, 2, 142-153		2012-02
One Step Synthesis of Optically Active Diazabicyclo[3.3.0]octanones or Diazabicyclo[4.3.0]nonanones by Asymmetric Conjugate Addition of Cyclic Hydrazine Heterocycles, 85, 5, 1045		2012-05
Highly Enantioselective Synthesis of Isoquinuclidine by Diels-Alder Reaction of 1,2-Dihydropyridine Utilizing Chiral Bisoxazoline-Cu(II) Complex Heterocycles, 86, 1, 203-217		2012-06
Asymmetric Synthesis of Isoquinuclidine by Diels-Alder Reaction of 1,2-Dihydropyridine and Chiral Dienophile Utilizing a Chiral Lewis Acid Heterocycles, 84, 1, 377-384		2012-06
CHIRAL PRIMARY AMINO SILYL ETHER ORGANOCATALYST FOR THE ENANTIOSELECTIVE DIELS-ALDER REACTION OF 1,2-DIHYDROPYRIDINES WITH AlDEHYDES Heterocycles, 86, 2		2012-08
Development of a Novel Method for Warfarin Synthesis via Lipase-Catalyzed Steroselective Michael Reaction Heterocycles, 87, 6, 1269-1278		2013-05
Enantioselective Diels–Alder Reaction of 1,2-Dihydropyridines with Aldehydes Using β-Amino Alcohol Organocatalyst J. Org. Chem., 79, 20, 9500-9511		2014-10
Chiral Primary Amino Amide Alcohol Organocatalyst for the Asymmetric Michael Addition of 4-Hydroxycoumarin with α,β-Unsaturated Ketones Heterocycles, 90, 2, 1124-1134		2015-07
Lipase-catalyzed domino Michael–aldol reaction of 2-methyl-1,3-cycloalkanedione and methyl vinyl ketone for the synthesis of bicyclic compounds Synth. commun., 46, 1, 46 - 54		2015-09
Silyloxy Amino Alcohol Organocatalyst for Enantioselective 1,3-Dipolar Cycloaddition of Nitrones to α,β-Unsaturated Aldehydes Eur. J. Org. Chem., 2015, 33, 7292-7300		2015-11
Chiral primary amino alcohol organobase catalysts for the asymmetric Diels–Alder reactions of anthrones with maleimides Tetrahedron: asymmetry, 26, 24, 1423-1429		2015-12
イミノ基により架橋した分解性ポリ(アルキルビニルエーテル)ゴムの合成 高分子論文集, 73, 73, 213-220		2016-03
Synthesis of Dibenzosiloles via Platinum-catalyzed Intramolecular Dehydrogenative Cyclization of 2-(Dialkylsilyl)biaryls Chemistry Letters, 45, 8, 857-859		2016-05
Simple Primary Amino Amide Organocatalyst for Enantioselective Aldol Reactions of Isatins with Ketones European Journal of Organic Chemistry, 2016, 22, 3748		2016-07
Site‐Selective Aliphatic C−H Silylation of 2‐Alkyloxazolines Catalyzed by Ruthenium Complexes CHEMCATCHEM, 8, 2202-2205		2016-07
Ruthenium-Catalysed Dehydrogenative C–H Borylation of Arenes with Pinacolborane Journal of Chemical Research, 40, 7, 393-396		2016-07
Rhodium(I)-Catalyzed Silylation of Aryl Iodides with Di(2-furyl)methylsilane Heterocycles, 95, 1, 152-157		2016-12
Simple primary β-amino alcohol catalyzed enantioselective Diels-Alder reaction of 3-hydroxy-2-pyridones Tetrahedron Letters, 57, 51, 5771		2016-12
Utilization of the Japanese peppermint herbal water byproduct of steam distillation as an antimicrobial agent Journal of Oleo Science, 67, 10, 1227-1233		2018-10
Unnatural tripeptide as highly enantioselective organocatalyst for asymmetric aldol reaction of isatins Tetrahedron Letters, 60, 5, 415-418		2018-12
Characteristics of Japanese Mint Extracts Obtained by Subcritical-water Treatment Food Science and Technology Research, 25, 5, 695-703		2019-01
Tripeptide-catalyzed Asymmetric Aldol Reaction of Trifluoromethylated Aromatic Ketones with Acetone Heterocycles, 99, 2, 841-847		2019-02
Preparation of monodisperse fully aromatic polyimide particles via the polycondensation of diethyl hexafluoroisopropylidenediphthalate with 4,4′-diaminodiphenylether in ethylene glycol Polymer Journal, 51, 405-412		2019-03
Tripeptide-Catalyzed Asymmetric Aldol Reaction Between α-ketoesters and Acetone Under Acidic Cocatalyst-Free Conditions Catalysts, 9, 6, 514		2019-06
Hydrodistillation by Solvent-Free Microwave Extraction of Fresh Japanese Peppermint (Mentha arvensis L.) Journal of Essential Oil Bearing Plants		2020-02
Conversion and Hydrothermal Decomposition of Major Components of Mint Essential Oil by Small-Scale Subcritical Water Treatment molecules, 25, 8, 1953		2020-04
トリペプチド触媒による活性化ケトン類の直接的不斉アルドール反応 有機合成化学協会誌, 78, 12, 1174-1183		2020-12
Organocatalyzed Asymmetric Aldol Reaction of α-Keto Amides with A Tripeptide Catalyst Synlett		2021-02
Chemical composition of essential oils obtained from Picea glehnii (F. Schmidt) Mast. grown in Hokkaido, Japan J. Essent. Oil Plant Comp., 2, 2, 99-103		2024-03
Tripeptide-Catalyzed Asymmetric Michael Addition Reaction of β-Nitrostyrenes with Cyclohexanone Synlett, 36, 3, 250-253		2024-04

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